SCHEMBL4767490

SCHEMBL4767490

[CH2]CC[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.47
ITGA2B P08514 10/20 0.47
TSHR P16473 1/20 0.47
CTSK P43235 5/20 0.45
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
TGM2 P21980 1/20 0.42
CTSS P25774 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767454 1.00 ITGB3 (0.47) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL27469415 0.87 CTSK (0.52) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL4916101 0.86 ITGB3 (0.50) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL4916104 0.86 ITGB3 (0.50) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL7453518 0.85 TSHR (0.49) ITGB3ITGA2BTSHRCTSKCTSS
SCHEMBL9103036 0.84 CTSK (0.52) ITGB3ITGA2BTSHRCTSKCTSS
SCHEMBL9103039 0.84 CTSK (0.52) ITGB3ITGA2BTSHRCTSKCTSS
SCHEMBL23845159 0.84 HRH2 (0.48) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL1706617 0.84 CTSK (0.54) ITGB3ITGA2BTSHRCTSKCTSL
SCHEMBL1707105 0.84 CTSK (0.54) ITGB3ITGA2BTSHRCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572678-A4 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS ELAN PHARM INC (US) 2008-05-07 EP claimed
EP-1572678-A2 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS Elan Pharmaceuticals, Inc. (US) 2005-09-14 EP claimed
EP-1501807-A1 SULFONYLQUINOXALONE ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ ANTAGONISTS Elan Pharmaceuticals, Inc. (US) 2005-02-02 EP claimed
WO-2004056319-A2 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS ELAN PHARMACEUTICALS INC. (US) 2004-07-08 WO claimed
WO-2003093245-A1 SULFONYLQUINOXALONE ACETAMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ ANTAGONISTS ELAN PHARMACEUTICALS, INC. (US) 2003-11-13 WO claimed