SCHEMBL4767640

SCHEMBL4767640

O=c1c2[nH]c(-c3cnn(-c4ccccc4)c3)cc2n(Cc2ccc(C(F)(F)F)cc2)c(=O)n1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 15/20 0.46
ADORA2A P29274 15/20 0.46
ADORA1 P30542 12/20 0.46
ADORA3 P0DMS8 8/20 0.41
GRM4 Q14833 1/20 0.40
CFTR P13569 1/20 0.39
PLK4 O00444 1/20 0.38
CDK2 P24941 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38
PLK3 Q9H4B4 1/20 0.38
CSNK1G3 Q9Y6M4 1/20 0.38
CTSK P43235 1/20 0.38
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769722 0.89 ADORA2B (0.48) ADORA2BADORA2AADORA1ADORA3GRM4
SCHEMBL4763685 0.85 ADORA2A (0.50) ADORA2BADORA2AADORA1ADORA3
SCHEMBL4771233 0.85 ADORA2B (0.52) ADORA2BADORA2AADORA1ADORA3PLK4
SCHEMBL4770636 0.83 ADORA2A (0.46) ADORA2BADORA2AADORA1ADORA3
SCHEMBL4763167 0.82 ADORA2B (0.55) ADORA2BADORA2AADORA1ADORA3PLK4
SCHEMBL4771316 0.82 ADORA2B (0.51) ADORA2BADORA2AADORA1ADORA3PLK4
SCHEMBL4769146 0.82 ADORA2B (0.48) ADORA2BADORA2AADORA1ADORA3
SCHEMBL4771327 0.82 ADORA2B (0.43) ADORA2BADORA2AADORA1ADORA3GRM4
SCHEMBL4767749 0.81 ADORA2A (0.44) ADORA2BADORA2AADORA1ADORA3
SCHEMBL4769743 0.80 ADORA2B (0.58) ADORA2BADORA2AADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed