SCHEMBL4768307

SCHEMBL4768307

CCCN(c1ncc2c(=O)c(C(N)=O)cn(-c3ccccc3)c2n1)n1ccnc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 17/20 0.47
PDE4A P27815 2/20 0.38
KCNH2 Q12809 1/20 0.38
NTRK1 P04629 3/20 0.36
KIT P10721 3/20 0.36
SRC P12931 3/20 0.36
FLT3 P36888 3/20 0.36
CAPN1 P07384 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772004 0.91 KCNH2 (0.41) CSF1RPDE4AKCNH2
SCHEMBL4773612 0.89 CSF1R (0.40) CSF1RPDE4AKCNH2
SCHEMBL4775827 0.86 CSF1R (0.59) CSF1RNTRK1KITSRCFLT3
SCHEMBL4777309 0.76 CSF1R (0.57) CSF1RNTRK1KITSRCFLT3
SCHEMBL4768934 0.74 CSF1R (0.45) CSF1RPDE4AKCNH2NTRK1KIT
SCHEMBL4775340 0.72 CSF1R (0.48) CSF1RPDE4AKCNH2NTRK1KIT
SCHEMBL4768393 0.72 CSF1R (0.47) CSF1RPDE4ANTRK1KITSRC
SCHEMBL3294019 0.71 CSF1R (0.75) CSF1RNTRK1KITSRCFLT3
SCHEMBL11016385 0.70 CSF1R (0.46) CSF1RPDE4AKCNH2
SCHEMBL3289880 0.69 CSF1R (0.56) CSF1RNTRK1KITSRCFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP claimed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO claimed
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP disclosed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO disclosed