SCHEMBL4768934

SCHEMBL4768934

CCCN(c1ncc2c(=O)c(C(N)=O)cn(-c3ccccc3)c2n1)C1CCNC1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 11/20 0.45
CHEK1 O14757 3/20 0.39
KCNH2 Q12809 2/20 0.39
RPS6KB1 P23443 1/20 0.38
SLC6A2 P23975 3/20 0.37
SLC6A4 P31645 3/20 0.37
SLC6A3 Q01959 2/20 0.36
NTRK1 P04629 1/20 0.35
KIT P10721 1/20 0.35
SRC P12931 1/20 0.35
FLT3 P36888 1/20 0.35
PDE4A P27815 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775792 0.94 SLC6A2 (0.38) CSF1RCHEK1KCNH2SLC6A2SLC6A4
SCHEMBL4775791 0.91 CSF1R (0.39) CSF1RKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL4777730 0.87 CSF1R (0.57) CSF1RNTRK1KITSRCFLT3
SCHEMBL4775340 0.80 CSF1R (0.48) CSF1RCHEK1KCNH2NTRK1KIT
SCHEMBL4768393 0.80 CSF1R (0.47) CSF1RNTRK1KITSRCFLT3
SCHEMBL4775794 0.78 CSF1R (0.55) CSF1RNTRK1KITSRCFLT3
SCHEMBL4572935 0.77 CSF1R (0.59) CSF1RNTRK1KITSRCFLT3
SCHEMBL4768307 0.74 CSF1R (0.47) CSF1RKCNH2NTRK1KITSRC
SCHEMBL4769014 0.71 CSF1R (0.42) CSF1RKCNH2PDE4A
SCHEMBL4793729 0.70 CSF1R (0.44) CSF1RNTRK1KITSRCFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP claimed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO claimed
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP disclosed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO disclosed