SCHEMBL4768355

SCHEMBL4768355

[C]C(CCNS(=O)(=O)c1ccc(Cl)cc1Cl)C(=O)NC1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.46
TRPV4 Q9HBA0 5/20 0.44
PPARG P37231 1/20 0.44
HSD11B1 P28845 3/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
PTGDR Q13258 2/20 0.42
PTGDR2 Q9Y5Y4 2/20 0.42
NPC1 O15118 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4136296 0.76 RAB9A (0.45) RAB9ATRPV4PPARGPTGDRPTGDR2
SCHEMBL4131127 0.75 RAB9A (0.39) RAB9ATRPV4PPARGPTGDRPTGDR2
SCHEMBL4132376 0.74 GAA (0.42) RAB9APPARGHSD11B1CA12CA1
SCHEMBL4131282 0.74 TRPV4 (0.44) RAB9ATRPV4PPARGHSD11B1PTGDR
SCHEMBL4152609 0.73 TRPV4 (0.40) RAB9ATRPV4CA12CA1CA2
SCHEMBL14605593 0.73 RAB9A (0.42) RAB9APPARGHSD11B1CA12CA1
SCHEMBL4777734 0.71 TRPV4 (0.55) TRPV4
SCHEMBL14606018 0.71 RAB9A (0.42) RAB9ATRPV4PPARGHSD11B1CA12
SCHEMBL4135553 0.71 CCR1 (0.40) RAB9APPARGHSD11B1PTGDRPTGDR2
SCHEMBL4136186 0.70 TRPV4 (0.39) RAB9ATRPV4PPARGHSD11B1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP claimed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO claimed