SCHEMBL4768622

SCHEMBL4768622

CCOCCSc1ccc(CC2CCN(C(C)=O)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CHRM2 P08172 6/20 0.44
GRIN2B Q13224 3/20 0.44
GRIN2A Q12879 2/20 0.44
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4773730 0.84 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AL3MBTL1CHRM2
SCHEMBL7512513 0.81 GRIN2B (0.46) ALDH1A1MEN1KMT2AGRIN2BGRIN2A
SCHEMBL4775580 0.79 CCR5 (0.54) ALDH1A1MEN1KMT2AL3MBTL1CYP2C9
SCHEMBL4779005 0.79 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL4771633 0.79 KCNH2 (0.47) CHRM2
SCHEMBL3031439 0.76 CHRM2 (0.61) CHRM2
SCHEMBL12801183 0.75 ALDH1A1 (0.43) ALDH1A1L3MBTL1CYP2C19
SCHEMBL4771768 0.74 CYP2C9 (0.43) ALDH1A1MEN1KMT2AL3MBTL1CHRM2
SCHEMBL4775057 0.73 SMN1; SMN2 (0.63) ALDH1A1MEN1KMT2ACHRM2GRIN2B
SCHEMBL14559864 0.73 MEN1 (0.56) ALDH1A1MEN1KMT2ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists TOBIRA THERAPEUTICS, INC. 2003-06-19 US disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists CCR5, CCR1, CCR3 ALDH1A1 3228/4885MEN1 2216/4885KMT2A 2421/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.