SCHEMBL4768985

SCHEMBL4768985

CCOC(=O)c1cn(CCO)ccc1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.46
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
CA9 Q16790 4/20 0.46
TSHR P16473 3/20 0.45
BAZ2B Q9UIF8 1/20 0.43
BAZ2A Q9UIF9 1/20 0.43
CA7 P43166 2/20 0.42
CA14 Q9ULX7 2/20 0.42
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 4/20 0.41
GAA P10253 4/20 0.41
GLA P06280 3/20 0.41
HPGD P15428 3/20 0.41
RAB9A P51151 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766475 0.85 TSHR (0.41) CA12CA1CA2CA9TSHR
SCHEMBL4773676 0.81 TSHR (0.50) CA12CA1CA2CA9TSHR
SCHEMBL31116594 0.80 TSHR (0.49) CA12CA1CA2CA9TSHR
SCHEMBL10314669 0.79 TSHR (0.53) CA12CA1CA2CA9TSHR
SCHEMBL4763560 0.78 CRHBP (0.38) CA12CA1CA2CA9TSHR
SCHEMBL4763568 0.75 CRHBP (0.36) CA12CA1CA2CA9TSHR
SCHEMBL21979601 0.75 BAZ2B (0.39) CA12CA1CA2CA9TSHR
SCHEMBL29209447 0.72 TSHR (0.41) CA12CA1CA2CA9TSHR
SCHEMBL30463107 0.72 TSHR (0.41) CA12CA1CA2CA9TSHR
SCHEMBL28840683 0.72 HTT (0.39) CA12CA1CA2CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309565-B1 HETEROCYCLIC MUTILIN ESTERS AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2008-04-09 EP disclosed
EP-1309565-A1 HETEROCYCLIC MUTILIN ESTERS AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002012199-A1 HETEROCYCLIC MUTILIN ESTERS AND THEIR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-14 WO disclosed