SCHEMBL4770075

SCHEMBL4770075

CC(C)(C)OC(=O)N1CCC[C@H]1N(c1ccc(F)c(Cl)c1)c1ccc(C#N)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PGR P06401 12/20 0.42
CYP2D6 P10635 12/20 0.42
CYP2C9 P11712 12/20 0.42
GPR119 Q8TDV5 1/20 0.42
ALDH1A1 P00352 1/20 0.41
AR P10275 3/20 0.39
LMNA P02545 2/20 0.39
TSHR P16473 2/20 0.39
POLQ O75417 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764174 0.87 MALT1 (0.43) PGRCYP2D6CYP2C9GPR119ALDH1A1
SCHEMBL4762739 0.86 ALDH1A1 (0.42) ALDH1A1LMNATSHRPOLQMEN1
SCHEMBL4762740 0.86 ALDH1A1 (0.42) ALDH1A1LMNATSHRPOLQMEN1
SCHEMBL4771661 0.85 ALDH1A1 (0.42) ALDH1A1LMNATSHRMEN1MAPT
SCHEMBL4771659 0.85 ALDH1A1 (0.42) ALDH1A1LMNATSHRMEN1MAPT
SCHEMBL4770053 0.84 TSHR (0.41) ALDH1A1LMNATSHRPOLQMEN1
SCHEMBL4770050 0.84 TSHR (0.41) ALDH1A1LMNATSHRPOLQMEN1
SCHEMBL4792059 0.84 ALDH1A1 (0.41) GPR119ALDH1A1LMNATSHRMEN1
SCHEMBL4792056 0.84 ALDH1A1 (0.41) GPR119ALDH1A1LMNATSHRMEN1
SCHEMBL4764121 0.84 APP (0.42) GPR119ALDH1A1LMNATSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881975-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-30 EP disclosed
WO-2006121218-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-11-16 WO disclosed