SCHEMBL4764121

SCHEMBL4764121

CC(C)(C)OC(=O)N1CCC[C@H]1N(c1ccc(S(C)(=O)=O)cc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
DRD2 P14416 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
SLC6A2 P23975 1/20 0.42
HRH2 P25021 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR7 P34969 1/20 0.42
DRD3 P35462 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR2B P41595 1/20 0.42
PSEN1 P49768 1/20 0.42
SLC6A3 Q01959 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4762740 0.88 ALDH1A1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4762739 0.88 ALDH1A1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4771659 0.87 ALDH1A1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4771661 0.87 ALDH1A1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4792056 0.85 ALDH1A1 (0.41) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4792059 0.85 ALDH1A1 (0.41) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4770075 0.84 PGR (0.42) GPR119MEN1KMT2AALDH1A1LMNA
SCHEMBL4766580 0.83 MEN1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4766576 0.83 MEN1 (0.42) APPHTR1AADRA2ADRD2ADRA2B
SCHEMBL4762745 0.82 GPR119 (0.45) APPHTR1AADRA2ADRD2ADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881975-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-30 EP disclosed
WO-2006121218-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-11-16 WO disclosed