SCHEMBL4770685

SCHEMBL4770685

CC(C)C[C@H](NC(=O)c1ccc(N2CCN(C(=O)O)CC2)cc1)C(=O)NCCCCNS(=O)(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.44
TRPV4 Q9HBA0 2/20 0.44
DRD2 P14416 3/20 0.43
DRD4 P21917 2/20 0.43
CTSL P07711 3/20 0.42
CTSS P25774 2/20 0.40
CCR1 P32246 4/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CAPN1 P07384 2/20 0.38
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
ADRA1A P35348 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4127687 0.91 SMN1; SMN2 (0.49) CTSKTRPV4DRD2DRD4CTSL
SCHEMBL13872529 0.91 SMN1; SMN2 (0.49) CTSKTRPV4DRD2DRD4CTSL
SCHEMBL4133648 0.82 CTSL (0.48) CTSKTRPV4CTSLCTSSCCR1
SCHEMBL13872567 0.82 CTSL (0.48) CTSKTRPV4CTSLCTSSCCR1
SCHEMBL4142303 0.77 CAPN1 (0.48) CTSKTRPV4CTSLCTSSCCR1
SCHEMBL4139657 0.75 CAPN1 (0.51) CTSKTRPV4CTSLCTSSCCR1
SCHEMBL4136044 0.74 TRPV4 (0.52) CTSKTRPV4CTSLCTSSCCR1
SCHEMBL4135455 0.74 TRPV4 (0.50) CTSKTRPV4CTSLCAPN1ALDH1A1
SCHEMBL4131282 0.74 TRPV4 (0.44) TRPV4CTSLCCR1CAPN1ALDH1A1
SCHEMBL4147709 0.74 TRPV4 (0.44) TRPV4CTSLCTSSCCR1CAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP claimed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO claimed