SCHEMBL4770852

SCHEMBL4770852

CCc1nnn(-c2ccccc2)c1C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.61
HTT P42858 1/20 0.51
ALDH1A1 P00352 4/20 0.49
TP53 P04637 3/20 0.48
ALOX12 P18054 1/20 0.48
NR4A3 Q92570 1/20 0.48
SLC5A1 P13866 1/20 0.45
SLC5A2 P31639 1/20 0.45
PPARG P37231 2/20 0.45
PPARA Q07869 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAOA P21397 1/20 0.41
GRN P28799 1/20 0.41
SORT1 Q99523 1/20 0.41
POLB P06746 2/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13543685 0.88 GPBAR1 (0.56) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL16697113 0.86 GPBAR1 (0.48) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL22897264 0.78 HTT (0.60) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL28824095 0.77 HTT (0.51) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL16004047 0.77 GPBAR1 (1.00) GPBAR1HTTALDH1A1NPC1RAB9A
SCHEMBL8621188 0.75 ALDH1A1 (0.49) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL27830568 0.74 POLB (0.48) HTTALDH1A1TP53ALOX12SMN1; SMN2
SCHEMBL4771914 0.74 HTT (0.64) GPBAR1HTTALDH1A1TP53ALOX12
SCHEMBL20028111 0.71 TP53 (0.66) HTTALDH1A1TP53ALOX12SLC5A1
SCHEMBL16697029 0.70 SLC5A1 (0.57) GPBAR1HTTALDH1A1TP53ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP disclosed