SCHEMBL4771460

SCHEMBL4771460

CCn1c(=O)c([N+](=O)[O-])c(C)n(CC2CC2)c1=O.c1cc2cc-2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
NPC1 O15118 1/20 0.39
MITF O75030 1/20 0.39
LMNA P02545 1/20 0.39
AGTR1 P30556 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TLR9 Q9NR96 1/20 0.39
KMT2A Q03164 2/20 0.38
GNRHR P30968 2/20 0.37
CYP1A2 P05177 1/20 0.37
PDE4A P27815 4/20 0.36
PDE4B Q07343 4/20 0.36
PDE4C Q08493 4/20 0.36
PDE4D Q08499 4/20 0.36
CFTR P13569 1/20 0.36
PDE5A O76074 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767817 0.89 PARG (0.38) PARGALDH1A1MAPTHTTNPC1
SCHEMBL4765596 0.81 ALDH1A1 (0.40) PARGALDH1A1MAPTHTTNPC1
SCHEMBL4762497 0.81 ALDH1A1 (0.43) ALDH1A1MAPTHTTNPC1MITF
SCHEMBL4771453 0.77 ADORA3 (0.44) ALDH1A1MAPTHTTNPC1MITF
SCHEMBL4767961 0.77 PDE4D (0.38) LMNANPSR1GNRHRPDE4APDE4B
SCHEMBL4771274 0.77 PDE5A (0.46) GNRHRPDE4APDE4BPDE4CPDE4D
SCHEMBL4057548 0.75 ALDH1A1 (0.44) ALDH1A1MAPTHTTNPC1MITF
SCHEMBL4767937 0.75 PDE4A (0.46) HTTKMT2AGNRHRPDE4APDE4B
SCHEMBL4765718 0.75 PDE4D (0.46) LMNANPSR1KMT2AGNRHRPDE4A
SCHEMBL4769379 0.75 ALDH1A1 (0.42) PARGALDH1A1MAPTLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed