SCHEMBL4771517

SCHEMBL4771517

Cn1cc(CCNc2cc(-c3cccnc3)nc(-c3ccccn3)n2)c2cc(Cl)ccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 2/20 0.40
CYP3A4 P08684 4/20 0.40
CDK2 P24941 1/20 0.40
CYP2C9 P11712 2/20 0.39
ROS1 P08922 3/20 0.39
SNCA P37840 1/20 0.39
TBXAS1 P24557 1/20 0.37
CLK4 Q9HAZ1 3/20 0.37
USP2 O75604 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PDE5A O76074 2/20 0.37
GPR39 O43194 1/20 0.37
CYP2A6 P11509 1/20 0.36
NR4A2 P43354 1/20 0.36
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2239882 0.91 PTGDR (0.42) PTGDRCYP3A4CDK2CYP2C9ROS1
SCHEMBL2239858 0.81 HPGD (0.57) CYP3A4CYP2C9SNCACLK4USP2
SCHEMBL4775435 0.80 HTR1A (0.40) PTGDRCYP3A4CYP2C9ROS1HDAC1
SCHEMBL2239769 0.80 CYP1A2 (0.49) PTGDRCYP3A4CDK2CYP2C9SNCA
SCHEMBL2242579 0.79 HTR6 (0.41) PTGDRCYP3A4CYP2C9ROS1CLK4
SCHEMBL2237203 0.78 CYP1A2 (0.48) PTGDRCYP3A4CYP2C9ROS1CLK4
SCHEMBL2237295 0.76 CYP2A6 (0.45) PTGDRCYP3A4CYP2C9CLK4USP2
SCHEMBL2238098 0.76 PTGDR (0.53) PTGDRCYP3A4CYP2C9CLK4USP2
SCHEMBL2240945 0.76 GBA1 (0.54) PTGDRCYP3A4CYP2C9CLK4CYP1A2
SCHEMBL2244237 0.76 CYP3A4 (0.47) CYP3A4CYP2C9CLK4USP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed