SCHEMBL4774131

SCHEMBL4774131

CCCN(c1ncc[nH]1)c1ccccc1[O]

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 7/20 0.37
HTR1A P08908 1/20 0.37
KCNA5 P22460 2/20 0.33
KCNH2 Q12809 1/20 0.33
CYP2D6 P10635 3/20 0.31
KCNE1 P15382 1/20 0.31
MTOR P42345 1/20 0.31
ADK P55263 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
F2RL1 P55085 2/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779621 0.90 TAAR1 (0.39) TAAR1HTR1ACYP2D6MTORADK
SCHEMBL4776714 0.78 TAAR1 (0.37) TAAR1HTR1AMTORADKNISCH
SCHEMBL4779370 0.72 TAAR1 (0.35) TAAR1HTR1AKCNA5KCNH2CYP2D6
SCHEMBL5350327 0.71 TAAR1 (0.34) TAAR1HTR1ACYP2D6CYP1A2CYP3A4
SCHEMBL5234870 0.70 HTT (0.51) TAAR1HTR1ACYP2D6MTORADK
SCHEMBL4977180 0.68 ALDH3A1 (0.40)
SCHEMBL4765598 0.68 HTT (0.40) TAAR1HTR1AKCNA5KCNH2CYP2D6
SCHEMBL4723517 0.67 TAAR1 (0.40) TAAR1HTR1AKCNA5KCNH2CYP2D6
SCHEMBL4721255 0.65 TAAR1 (0.44) TAAR1HTR1AKCNA5CYP2D6KCNE1
SCHEMBL6741597 0.65 TGFBR1 (0.34) TAAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed