SCHEMBL4774546

SCHEMBL4774546

Brc1cccc(Nc2ncc3cc(-c4cnn(CC5OCCO5)c4)ccc3n2)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 3/20 0.44
BRAF P15056 5/20 0.42
MAP3K5 Q99683 2/20 0.42
DGAT1 O75907 1/20 0.42
KDR P35968 2/20 0.40
AURKB Q96GD4 1/20 0.39
MAP4K3 Q8IVH8 1/20 0.39
IKBKE Q14164 1/20 0.39
TBK1 Q9UHD2 1/20 0.39
CDK1 P06493 1/20 0.38
DDR2 Q16832 3/20 0.37
AXL P30530 1/20 0.37
TYRO3 Q06418 1/20 0.37
MERTK Q12866 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
CCNA1 P78396 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4354964 0.80 EGFR (0.46) KDRAURKBIKBKETBK1
SCHEMBL25882292 0.68 SCN9A (0.51) BRAFDDR2
SCHEMBL13336325 0.66 MAP4K1 (0.45) MAP4K1KDRTBK1CDK1CCNA2
SCHEMBL4358324 0.66 PIK3CA (0.42) IKBKETBK1
SCHEMBL5909044 0.66 FBP1 (0.58) BRAFKDRCDK1
SCHEMBL12725589 0.66 MAPK10 (0.55) MAP4K1MAP4K3CCNA2CDK2
SCHEMBL1632778 0.65 MAPK10 (0.53) MAP4K1CCNA2CDK2
SCHEMBL2741577 0.65 BRAF (0.60) MAP4K1BRAFMAP3K5DGAT1KDR
SCHEMBL5495505 0.65 ADRB2 (0.58) BRAFMAP3K5DGAT1KDRAURKB
SCHEMBL13362987 0.65 MAP3K5 (0.62) BRAFMAP3K5KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009078-A2 4,6-DL- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed