SCHEMBL4775229

SCHEMBL4775229

CCOC(=O)COc1ccc(O)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
L3MBTL1 Q9Y468 3/20 0.57
TDP1 Q9NUW8 2/20 0.57
ADRB3 P13945 2/20 0.56
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
HPGD P15428 1/20 0.50
CASP1 P29466 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TSHR P16473 2/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
MAPK1 P28482 1/20 0.49
ESR1 P03372 1/20 0.49
CASP3 P42574 1/20 0.48
CASP7 P55210 1/20 0.48
CASP9 P55211 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29369910 0.86 TDP1 (0.74) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL1694924 0.86 TDP1 (0.74) ALDH1A1L3MBTL1TDP1KDM4ETSHR
SCHEMBL2007090 0.86 ALDH1A1 (0.56) ALDH1A1ADRB3KDM4EMEN1HPGD
SCHEMBL1549799 0.84 ESR1 (0.61) ALDH1A1KDM4EMEN1HPGDCASP1
SCHEMBL1815302 0.84 ALDH1A1 (0.56) ALDH1A1L3MBTL1TDP1ADRB3KDM4E
SCHEMBL4303747 0.84 ALDH1A1 (0.65) ALDH1A1L3MBTL1TDP1KDM4EMEN1
SCHEMBL3531540 0.84 ALDH1A1 (0.56) ALDH1A1L3MBTL1TDP1ADRB3KDM4E
SCHEMBL2031260 0.83 ALDH1A1 (0.50) ALDH1A1ADRB3KDM4EMEN1HPGD
SCHEMBL4773036 0.82 ALDH1A1 (0.58) ALDH1A1L3MBTL1TDP1ADRB3KDM4E
SCHEMBL2007531 0.82 ALDH1A1 (0.54) ALDH1A1L3MBTL1TDP1ADRB3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937647-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II Inpharmatica Limited (GB) 2008-07-02 EP disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed
WO-2007036727-A1 CONDENSED PYRAZOLE DERIVATIVES AS PPAR AGONISTS II INPHARMATICA LIMITED (GB) 2007-04-05 WO disclosed