SCHEMBL47762

SCHEMBL47762

COCCOC(=O)C1(OCCOC)CCC(c2cc(NCOCC[Si](C)(C)C)n3ncc(-c4cnn(-c5ccccc5)c4)c3n2)CC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCNA1 P78396 1/20 0.38
TYK2 P29597 1/20 0.35
GRM4 Q14833 3/20 0.34
DGAT1 O75907 1/20 0.34
TTK P33981 3/20 0.33
RIPK2 O43353 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21073 0.89 GRM4 (0.34) CHEK1CCNA2CDK2CCNA1TYK2
SCHEMBL30524 0.86 GRM4 (0.32) GRM4
SCHEMBL21078 0.83 GRM4 (0.34) CHEK1CCNA2CDK2CCNA1TYK2
SCHEMBL40556 0.83 HSD17B10 (0.33)
SCHEMBL19684 0.83 GRM4 (0.32) GRM4DGAT1
SCHEMBL15031440 0.82 JAK2 (0.31)
SCHEMBL15006969 0.82 JAK2 (0.31)
SCHEMBL15006968 0.82 JAK2 (0.31)
SCHEMBL15007081 0.82 GRM4 (0.34) CHEK1CCNA2CDK2CCNA1TYK2
SCHEMBL19940 0.81 GRM4 (0.32) GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027234-A1 FUSED TRICYCLIC INHIBITORS OF MAMMALIAN TARGET OF RAPAMYCIN SCHERING CORPORATION (US) 2012-03-01 WO disclosed