SCHEMBL4776364

SCHEMBL4776364

COC(=O)c1sc(I)cc1NC1CCOC1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
PDE1B Q01064 4/20 0.33
PDE1C Q14123 4/20 0.33
PDE1A P54750 2/20 0.33
HSP90AA1 P07900 2/20 0.33
HSP90AB1 P08238 2/20 0.33
HSP90B1 P14625 2/20 0.33
PDCD1 Q15116 2/20 0.33
CD274 Q9NZQ7 2/20 0.33
TRAP1 Q12931 1/20 0.33
LRRK2 Q5S007 2/20 0.33
HPGD P15428 1/20 0.33
FASN P49327 1/20 0.32
OPRK1 P41145 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731070 0.92 LRRK2 (0.38) HPGDSKDM4EHTTATMLRRK2
SCHEMBL12444721 0.80 ALDH1A1 (0.36) KDM4EHTTATMHPGDSMN1; SMN2
SCHEMBL4730428 0.77 SMN1; SMN2 (0.52) KDM4EHTTHPGDSMN1; SMN2KMT2A
SCHEMBL2430706 0.74 PTGER4 (0.46) KDM4EHTTATMHPGDSMN1; SMN2
SCHEMBL11922640 0.73 CFTR (0.37) KDM4EHSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL2874896 0.72 KDM4E (0.63) KDM4EHTTATMHPGDKMT2A
SCHEMBL1963295 0.71 CYP2E1 (0.39) HPGDSKDM4EHTTATMLRRK2
SCHEMBL669499 0.71 ACACB (0.35) KDM4EHTTATMLRRK2OPRK1
SCHEMBL12945315 0.70 RAF1 (0.43)
SCHEMBL12945290 0.70 RAF1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed
WO-2008043791-A2 THIOPHENE DERIVATIVES FOR TREATING HEPATITIS C SMITHKLINE BEECHAM CORPORATION (US) 2008-04-17 WO disclosed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed