SCHEMBL4777264

SCHEMBL4777264

Cc1onc(CO)c1CCNCc1csc(NC(=O)NCc2cccc(F)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 15/20 0.49
ROCK1 Q13464 15/20 0.49
EPHX2 P34913 1/20 0.41
ATG4B Q9Y4P1 1/20 0.40
SGK1 O00141 1/20 0.38
AKT1 P31749 1/20 0.38
GSK3B P49841 1/20 0.38
LIMK1 P53667 1/20 0.38
TNK2 Q07912 1/20 0.38
DMPK Q09013 1/20 0.38
MYLK Q15746 1/20 0.38
CDC42BPA Q5VT25 1/20 0.38
MAPK1 P28482 1/20 0.37
THRB P10828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4725210 0.99 ROCK2 (0.49) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL4777272 0.86 ROCK2 (0.50) ROCK2ROCK1EPHX2ATG4BSGK1
Hydrochloric Acid SCHEMBL4725212 0.86 ROCK2 (0.49) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL354195 0.85 ROCK1 (0.54) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL353543 0.82 ROCK2 (0.62) ROCK2ROCK1EPHX2ATG4B
SCHEMBL352833 0.80 ROCK2 (0.49) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL3656133 0.80 ROCK2 (0.60) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL10237499 0.79 ROCK2 (0.61) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL354019 0.79 ROCK1 (0.68) ROCK2ROCK1EPHX2ATG4BSGK1
SCHEMBL354438 0.78 ROCK1 (0.49) ROCK2ROCK1EPHX2ATG4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008011191-A1 ANTIBACTERIAL HETEROCYCLIC UREAS REPLIDYNE, INC. (US) 2008-01-24 WO disclosed