SCHEMBL4778154

SCHEMBL4778154

NC(C=O)C(c1ccc(Br)s1)N1CCN(C(=O)c2c(Cl)ncc(F)c2Cl)CC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.34
BCR P11274 2/20 0.34
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KMT2A Q03164 2/20 0.32
MET P08581 1/20 0.32
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772508 0.79 CYP3A4 (0.36) MET
SCHEMBL4778149 0.75 HDAC8 (0.39) ABL1BCRRECQLHSD17B10
SCHEMBL4776893 0.73 SCD (0.39) ABL1BCRRECQLHSD17B10KMT2A
SCHEMBL4837579 0.72 SCD (0.38) RECQLHSD17B10KMT2AKDM4E
SCHEMBL4779060 0.66 CYP1A2 (0.42) KMT2AALDH1A1LMNAKDM4E
SCHEMBL4794759 0.66 DPP4 (0.43) KMT2AALDH1A1LMNAKDM4EMEN1
SCHEMBL4779485 0.65 DPP8 (0.35)
SCHEMBL4770020 0.64 AKT1 (0.52) KMT2AMEN1
SCHEMBL4779334 0.64
SCHEMBL4779275 0.63 HDAC8 (0.65) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996550-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES Novartis AG (CH) 2008-12-03 EP claimed
WO-2007038459-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES NOVARTIS AG (CH) 2007-04-05 WO claimed