SCHEMBL4778736

SCHEMBL4778736

Cc1cccc(C)c1Sc1[c]cccc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
ACHE P22303 1/20 0.35
SCN4A P35499 4/20 0.33
CYP2A6 P11509 2/20 0.31
ALDH1A1 P00352 2/20 0.31
AR P10275 2/20 0.31
CYP1A2 P05177 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16053808 0.88 ACHE (0.41) ACHE
SCHEMBL467564 0.84 HAO1 (0.40) TSHRACHEALDH1A1ARCA1
SCHEMBL2423602 0.78
SCHEMBL1783489 0.72 CYP2A6 (0.47) TSHRACHESCN4ACYP2A6ALDH1A1
SCHEMBL483135 0.72 MAPT (0.43) TSHRACHEALDH1A1CYP1A2
SCHEMBL7636503 0.72 HTR1A (0.39) ACHEALDH1A1
SCHEMBL9334108 0.72 TSHR (0.31) TSHRACHESCN4A
SCHEMBL3717937 0.71 HTR1A (0.42) CYP1A2
SCHEMBL237661 0.70 HPGD (0.38) ALDH1A1
SCHEMBL9488226 0.69 HAO1 (0.47) TSHRACHESCN4ACYP2A6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436271-B1 PHENYL-PIPERAZINE DERIVATIVES AS SEROTONIN REUPTAKE INHIBITORS LUNDBECK & CO AS H (DK) 2008-02-20 EP claimed
EP-1089963-B1 HYDROXAMIC ACID DERIVATIVES AS INHIBITORS OF THE PRODUCTION OF HUMAN CD23 AND OF THE TNF RELEASE SMITHKLINE BEECHAM PLC (GB) 2004-06-16 EP claimed
US-6458779-B1 TREATMENT OF CONDITIONS ASSOCIATED WITH EXCESS PRODUCTION OF SOLUBLE CD23 (S-CD23) SUCH AS AUTOIMMUNE DISEASE AND ALLERGY. THE COMPOUNDS OF THE INVENTION ARE ALSO INHIBITORS OF THE RELEASE OF TUMOUR NECROSIS FACTOR (TNF). SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-01 US claimed