SCHEMBL4779574

SCHEMBL4779574

COc1cc2ncnc(N3CCCC3)c2cc1O

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.63
BACE1 P56817 9/20 0.63
PDE10A Q9Y233 1/20 0.61
ENPP1 P22413 7/20 0.61
AURKA O14965 1/20 0.58
PDGFRB P09619 1/20 0.57
PDE3A Q14432 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779400 0.99 ACHE (0.61) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL4726710 0.97 ENPP1 (0.65) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL3873291 0.88 ACHE (0.78) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL5518977 0.87 ACHE (0.76) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL13529592 0.84 ACHE (0.80) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL11882354 0.82 ACHE (0.88) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL23762347 0.81 ENPP1 (0.85) ACHEBACE1PDE10AENPP1AURKA
SCHEMBL29055014 0.81 ACHE (0.64) ACHEBACE1ENPP1AURKAPDGFRB
SCHEMBL25656495 0.81 ENPP1 (0.59) ACHEBACE1PDE10AENPP1AURKA
Hydrochloric Acid SCHEMBL30079993 0.80 ENPP1 (0.84) ACHEBACE1PDE10AENPP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed