SCHEMBL4779653

SCHEMBL4779653

FC(F)(F)c1ccc(-c2ccccc2)cc1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.58
RXRB P28702 1/20 0.58
RXRG P48443 1/20 0.58
KIF11 P52732 6/20 0.54
NOTUM Q6P988 1/20 0.46
CYP11B2 P19099 2/20 0.45
AR P10275 5/20 0.42
PTPN1 P18031 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
S1PR1 P21453 1/20 0.41
LDHA P00338 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28222645 1.00 RXRA (0.58) RXRARXRBRXRGKIF11NOTUM
SCHEMBL28231443 0.90 RXRA (0.54) RXRARXRBRXRGKIF11NOTUM
SCHEMBL27638533 0.83 S1PR1 (0.52) RXRARXRBRXRGKIF11AR
SCHEMBL6120541 0.83 KIF11 (0.69) KIF11CYP11B2
SCHEMBL4636314 0.81 S1PR1 (0.60) RXRARXRBRXRGKIF11NOTUM
SCHEMBL1041026 0.81 ESR2 (0.52) RXRARXRBRXRGKIF11CYP11B2
SCHEMBL1042573 0.81 NOTUM (0.50) RXRARXRBRXRGKIF11NOTUM
SCHEMBL1040661 0.81 KIF11 (0.48) RXRARXRBRXRGKIF11NOTUM
SCHEMBL31570062 0.81 KIF11 (0.57) RXRARXRBRXRGKIF11CYP11B2
SCHEMBL3785824 0.81 KIF11 (0.57) RXRARXRBRXRGKIF11CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050075324-A1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2005-04-07 US claimed
CN-109239816-A Laminated film, and display device including the same 三星电子株式会社 2019-01-18 CN disclosed
CN-103254250-B Ferrocenyl pyridine cyclic Pd-N heterocyclic carbene compound as well as preparation method and application thereof UNIV LUOYANG NORMAL 2015-06-10 CN disclosed
US-7368462-B1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2008-05-06 US disclosed
US-20080058423-A1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY 2008-03-06 US disclosed
WO-2008001160-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO disclosed
US-7304065-B2 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2007-12-04 US disclosed
US-20060247239-A1 Melanin concentrating hormone antagonists HU XIUFENG E 2006-11-02 US disclosed
EP-1667958-A2 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2006-06-14 EP disclosed
WO-2005033063-A2 MELANIN CONCENTRATING HORMONE ANTAGONISTS THE PROCTER & GAMBLE COMPANY (US) 2005-04-14 WO disclosed
US-20050075324-A1 Melanin concentrating hormone antagonists THE PROCTER & GAMBLE COMPANY (US) 2005-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080058423-A1 Melanin concentrating hormone antagonists MCHR1, MCHR2, MC4R RXRA 1066/4885RXRB 1075/4885RXRG 777/4885
US-20050075324-A1 Melanin concentrating hormone antagonists MCHR1, MCHR2, MC1R RXRA 1395/4885RXRB 1565/4885RXRG 1073/4885
US-20060247239-A1 Melanin concentrating hormone antagonists MCHR1, MCHR2, MC1R RXRA 1395/4885RXRB 1565/4885RXRG 1073/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.