SCHEMBL4779958

SCHEMBL4779958

CCOC(=O)c1cc[nH]c1-c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.56
MAPT P10636 4/20 0.56
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51
PRKCZ Q05513 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ADORA3 P0DMS8 1/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HTT P42858 1/20 0.45
CACNA1D Q01668 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3493726 0.80 TSHR (0.58) MAPTGAARAB9ASMN1; SMN2KMT2A
SCHEMBL9979815 0.79 AR (0.64) ARMAPTGAARAB9APRKCZ
SCHEMBL276323 0.78 AR (0.56) ARMAPTGAARAB9APRKCZ
SCHEMBL30741033 0.77 GCGR (0.56) ARMAPTSMN1; SMN2ADORA3KMT2A
SCHEMBL28362521 0.77 KCNJ1 (0.64) ARMAPTGAARAB9APRKCZ
SCHEMBL7640668 0.77 MAPT (0.57) ARMAPTGAARAB9APRKCZ
SCHEMBL30740871 0.76 ALDH1A1 (0.49) MAPTGAARAB9ASMN1; SMN2ADORA3
SCHEMBL16043087 0.76 AR (0.60) ARMAPTGAARAB9APRKCZ
SCHEMBL7439474 0.76 AR (0.60) ARMAPTGAARAB9APRKCZ
SCHEMBL30741042 0.76 GCGR (0.55) ARMAPTGAARAB9APRKCZ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957078-A2 PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING CANCER THROUGH INHIBITION OF AURORA KINASE Bayer Healthcare, LLC (US) 2008-08-20 EP disclosed
WO-2007064932-A2 PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING CANCER THROUGH INHIBITION OF AURORA KINASE BAYER HEALTHCARE LLC. (US) 2007-06-07 WO disclosed