SCHEMBL4780351

SCHEMBL4780351

CCOc1ccc(-c2cncc(F)c2)cc1CNC1CCC(N(C)C(=O)OC(C)(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.39
ADORA2B P29275 2/20 0.39
IRAK4 Q9NWZ3 2/20 0.39
NPBWR1 P48145 1/20 0.36
MCHR1 Q99705 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
ABL1 P00519 1/20 0.35
KAT6A Q92794 1/20 0.35
KAT8 Q9H7Z6 1/20 0.35
GRIN2B Q13224 3/20 0.35
DYRK1A Q13627 5/20 0.34
WNT1 P04628 1/20 0.34
KCNH2 Q12809 2/20 0.34
CYP2D6 P10635 1/20 0.34
GSK3B P49841 2/20 0.34
GPR119 Q8TDV5 1/20 0.34
GRIN1 Q05586 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
CTPS1 P17812 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734472 0.92 KCNH2 (0.41) ADORA2AADORA2BIRAK4ABL1KAT6A
SCHEMBL12678651 0.92 KCNH2 (0.41) ADORA2AADORA2BIRAK4ABL1KAT6A
SCHEMBL12678417 0.87 NPBWR1 (0.38) IRAK4NPBWR1MCHR1PPARDABL1
SCHEMBL12690573 0.84 NPBWR1 (0.39) NPBWR1MCHR1PPARDPPARAGPR119
SCHEMBL12678471 0.83 PPARD (0.38) NPBWR1MCHR1PPARDPPARAGPR119
SCHEMBL12680623 0.83 PPARD (0.38) NPBWR1MCHR1PPARDPPARAGPR119
SCHEMBL12680480 0.83 GPR119 (0.40) NPBWR1MCHR1KAT6AKAT8GPR119
SCHEMBL12678379 0.83 NPBWR1 (0.38) NPBWR1MCHR1PPARDABL1KAT6A
SCHEMBL12678648 0.82 MEN1 (0.36) ABL1KAT6AKAT8GRIN2BDYRK1A
SCHEMBL4730577 0.82 MEN1 (0.36) ABL1KAT6AKAT8GRIN2BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008057497-A2 SMALL ORGANIC MOLECULE REGULATORS OF CELL PROLIFERATION CURIS, INC. (US) 2008-05-15 WO disclosed