SCHEMBL4780802

SCHEMBL4780802

NC(=O)N1CC=Cc2ccncc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 1/20 0.37
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
SCN4A P35499 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
CYP11B2 P19099 14/20 0.34
SIRT3 Q9NTG7 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
NAMPT P43490 1/20 0.32
F7 P08709 1/20 0.32
F3 P13726 1/20 0.32
SARM1 Q6SZW1 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
SIRT6 Q8N6T7 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
SIRT5 Q9NXA8 1/20 0.32
SIRT4 Q9Y6E7 1/20 0.32
HDAC3 O15379 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoquinoline SCHEMBL28191779 0.81 LMNA (0.40) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL1286806 0.77 LMNA (0.55) P2RX4LMNATSHRMAPK1SCN4A
Hydrochloric Acid SCHEMBL28145471 0.76 LMNA (0.53) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL5823517 0.73 KDM4E (0.32) P2RX4CYP11B2TDP1
SCHEMBL15083805 0.73 P2RX4 (0.36) P2RX4HDAC3HDAC1HDAC2HDAC6
SCHEMBL1836164 0.69 PARP1 (0.36) LMNATSHRMAPK1SCN4ASCN5A
SCHEMBL30511570 0.69 PARP1 (0.36) LMNATSHRMAPK1SCN4ASCN5A
SCHEMBL16671338 0.69 PARP1 (0.36) LMNATSHRMAPK1SCN4ASCN5A
Isoquinoline SCHEMBL28075529 0.68 P2RX4 (0.38) P2RX4LMNATSHRMAPK1SCN4A
SCHEMBL28778878 0.67 LMNA (0.40) P2RX4LMNATSHRMAPK1SCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008001134-A1 1,2,3,8,9,9A-HEXAHYDRO-7H-BENZO(DE)-1,7-NAPHTHYRIDIN-7-ONE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2008-01-03 WO disclosed