Isoquinoline

Isoquinoline

SCHEMBL28075529

O=C(O)N1CC=Cc2ccccc21.c1ccc2cnccc2c1

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 6/20 0.38
IMPDH2 P12268 2/20 0.36
CYP3A4 P08684 1/20 0.34
TRPV1 Q8NER1 3/20 0.33
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ROCK2 O75116 2/20 0.32
ROCK1 Q13464 1/20 0.32
STAT3 P40763 1/20 0.32
MAPK1 P28482 2/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
SCN4A P35499 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
MEN1 O00255 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isoquinoline SCHEMBL28191779 0.89 LMNA (0.40) P2RX4IMPDH2TRPV1HDAC3HDAC1
SCHEMBL29376182 0.83 P2RX4 (0.44) P2RX4MAPK1LMNATSHRSCN4A
SCHEMBL3375661 0.83 P2RX4 (0.44) P2RX4MAPK1LMNATSHRSCN4A
SCHEMBL5823517 0.81 KDM4E (0.32) P2RX4CYP3A4MEN1KMT2A
Quinoline SCHEMBL28157604 0.80 ALDH1A1 (0.44) P2RX4CYP3A4TRPV1MAPK1LMNA
Isoquinoline SCHEMBL28191817 0.79 CA12 (0.33) P2RX4CYP3A4ROCK2ROCK1LMNA
Indole SCHEMBL28214491 0.75 TRPA1 (0.45) P2RX4MAPK1LMNATSHRSCN4A
Isoquinoline SCHEMBL28183569 0.75 HTT (0.33) P2RX4HTT
Isoquinoline SCHEMBL11346369 0.72 IMPDH2 (0.53) IMPDH2CYP3A4TRPV1ROCK2ROCK1
SCHEMBL3241414 0.71 P2RX4 (0.42) P2RX4MAPK1LMNATSHRSCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008540-A Heterocyclic aromatic acid ester type podophyllotoxin derivatives with anti-tumor activity as well as preparation method and application 遵义医学院 2016-10-12 CN claimed