SCHEMBL4781129

SCHEMBL4781129

C[C@H]1CC[C@H](C(=O)N(c2cc(-c3ccc(-c4cn5ccccc5n4)cc3)sc2C(=O)O)C2CCOCC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.42
KDM4E B2RXH2 11/20 0.41
SMN1; SMN2 Q16637 8/20 0.41
ALDH1A1 P00352 8/20 0.41
HPGD P15428 6/20 0.41
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
HSD17B10 Q99714 3/20 0.39
MAPT P10636 2/20 0.39
RAB9A P51151 7/20 0.36
NPC1 O15118 5/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 2/20 0.36
EPHX2 P34913 1/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GFER P55789 4/20 0.35
USP2 O75604 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781136 1.00 FASN (0.42) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4776126 0.90 FASN (0.41) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4776116 0.90 FASN (0.41) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4725812 0.87 FASN (0.41) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4725816 0.87 FASN (0.41) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4776100 0.87 SMN1; SMN2 (0.43) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL4776105 0.87 SMN1; SMN2 (0.43) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL4152130 0.86 PTGS1 (0.45) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL4152135 0.86 PTGS1 (0.45) FASNKDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL2244516 0.84 CYP2E1 (0.40) KDM4EALDH1A1HSD17B10MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO claimed
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed