SCHEMBL4782645

SCHEMBL4782645

NC(=O)c1ccc(F)nc1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.44
PARP1 P09874 5/20 0.43
CDC7 O00311 2/20 0.42
IKBKB O14920 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
BTK Q06187 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
DHODH Q02127 1/20 0.39
MAP2K3 P46734 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6616377 0.81 BCAT2 (0.47) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL29002505 0.79 KDM4E (0.53) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL4504523 0.79 JAK2 (0.49) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL1533665 0.76 PARP1 (0.54) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL30017135 0.75 KDM4E (0.40) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL28639243 0.75 KDM4E (0.40) BCAT2MEN1KMT2AKDM4EALDH1A1
SCHEMBL30733977 0.74 DGAT1 (0.42) MEN1KMT2AKDM4EALDH1A1PARP1
SCHEMBL2762235 0.74 DGAT1 (0.42) MEN1KMT2AKDM4EALDH1A1PARP1
SCHEMBL30641935 0.74 DGAT1 (0.42) MEN1KMT2AKDM4EALDH1A1PARP1
Benzoic Acid SCHEMBL28961466 0.73 TSHR (0.45) BCAT2MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed
CN-1176908-C Process for producing pyridine derivate - 2004-11-24 CN disclosed
CN-1297887-A Process for producing pyridine derivate HOFFMANN LA ROCHE (CH) 2001-06-06 CN disclosed