SCHEMBL4782980

SCHEMBL4782980

NCCNc1nc(-c2cccc(O)c2)nc(N2CCc3ccccc3C2CO)n1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.44
ESR2 Q92731 3/20 0.35
ESR1 P03372 2/20 0.35
IDH1 O75874 1/20 0.35
CSNK1D P48730 1/20 0.35
PFKFB3 Q16875 1/20 0.34
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
HTR1A P08908 1/20 0.33
GPR68 Q15743 1/20 0.33
GBA1 P04062 1/20 0.32
KDM6B O15054 1/20 0.32
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4855287 0.93 PIK3CA (0.44) PIK3CAESR2ESR1IDH1PFKFB3
SCHEMBL4784449 0.86 PIK3CA (0.49) PIK3CAPIK3CBPIK3CG
SCHEMBL4784144 0.84 IDH1 (0.42) PIK3CAESR2ESR1IDH1PFKFB3
SCHEMBL4784052 0.82 PIK3CA (0.38) PIK3CAESR2ESR1IDH1PFKFB3
SCHEMBL4785148 0.82 ESR1 (0.42) PIK3CAESR2ESR1PFKFB3PRMT5
SCHEMBL4782612 0.81 IDH1 (0.41) PIK3CAESR2ESR1IDH1PFKFB3
SCHEMBL4781508 0.81 PIK3CA (0.42) PIK3CAESR2ESR1
SCHEMBL4784160 0.80 PIK3CA (0.42) PIK3CAESR2ESR1PFKFB3
SCHEMBL4785552 0.80 PIK3CA (0.42) PIK3CAESR2ESR1PFKFB3PIK3CB
SCHEMBL4784501 0.80 AOC3 (0.38) PIK3CAESR2ESR1IDH1PFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed