SCHEMBL4784449

SCHEMBL4784449

OCC1c2ccccc2CCN1c1nc(NCCN2CCOCC2)nc(-c2cccc(O)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.49
MTOR P42345 3/20 0.46
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
USP2 O75604 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FYN P06241 1/20 0.39
PIK3CG P48736 3/20 0.39
PIK3CB P42338 2/20 0.39
PIK3CD O00329 1/20 0.39
TLR9 Q9NR96 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4855287 0.88 PIK3CA (0.44) PIK3CA
SCHEMBL4782980 0.86 PIK3CA (0.44) PIK3CAPIK3CGPIK3CB
SCHEMBL4785203 0.84 KDR (0.42) PIK3CAMTORPIK3CGPIK3CBPIK3CD
SCHEMBL4782724 0.83 PIK3CA (0.57) PIK3CAMTORPIK3CGPIK3CBPIK3CD
SCHEMBL4784452 0.83 PIK3CA (0.50) PIK3CAMTORMEN1KMT2ALMNA
SCHEMBL4784144 0.80 IDH1 (0.42) PIK3CAMTORMAPTALDH1A1MAPK1
SCHEMBL4784015 0.78 HTR2A (0.44) PIK3CAMTORMEN1KMT2ALMNA
SCHEMBL4783015 0.78 PIK3CA (0.48) PIK3CAMTORPIK3CG
SCHEMBL4784052 0.78 PIK3CA (0.38) PIK3CAMTORLMNACYP1A2CYP3A4
SCHEMBL4785148 0.78 ESR1 (0.42) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed