SCHEMBL4784015

SCHEMBL4784015

OCCN1CCN(c2nc(-c3cccc(O)c3)nc(N3CCc4ccccc4C3CO)n2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
PIK3CA P42336 10/20 0.42
KDM4E B2RXH2 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
USP2 O75604 1/20 0.40
TP53 P04637 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MTOR P42345 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 2/20 0.38
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781508 0.93 PIK3CA (0.42) HTR2APIK3CAMEN1KMT2AMTOR
SCHEMBL4783923 0.92 HRH4 (0.43) PIK3CASMN1; SMN2MTORCYP2C19ESR1
SCHEMBL4782297 0.90 PIK3CA (0.43) PIK3CAMTORESR1ESR2ADORA3
SCHEMBL4784640 0.88 ADORA3 (0.43) PIK3CAMTORESR1ESR2ADORA3
SCHEMBL4784804 0.88 ESR1 (0.41) PIK3CAMTORESR1ESR2ADORA3
SCHEMBL4784088 0.88 PIK3CA (0.43) PIK3CAKMT2AALDH1A1MTORESR1
SCHEMBL4782788 0.87 PIK3CA (0.42) PIK3CAALDH1A1MAPTTSHRSMN1; SMN2
SCHEMBL4782724 0.87 PIK3CA (0.57) PIK3CAMTOR
SCHEMBL4884094 0.87 PIK3CA (0.44) PIK3CAMTORESR1ESR2
SCHEMBL4784160 0.87 PIK3CA (0.42) PIK3CAMTORESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed