SCHEMBL4784586

SCHEMBL4784586

Cc1noc2ccnc(O)c12

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.36
ALDH1A1 P00352 4/20 0.33
ALOX15 P16050 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
LMNA P02545 2/20 0.32
USP2 O75604 1/20 0.32
GFER P55789 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP2A6 P11509 1/20 0.31
HTT P42858 2/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3195416 0.71 KCNA5 (0.46) ALDH1A1ALOX15MAPTCYP1A2CYP3A4
SCHEMBL4784582 0.67 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTCYP1A2LMNA
SCHEMBL25669745 0.65 CYP1A2 (0.41) DRD1ALDH1A1L3MBTL1MAPTCYP1A2
SCHEMBL8404487 0.65 CYP1A2 (0.41) ALDH1A1MAPTCYP1A2LMNACYP2C19
SCHEMBL24302564 0.64 MAOA (0.39) MAPTCYP1A2LMNAGFERCYP2C9
SCHEMBL10200850 0.64 ALDH1A1 (0.45) ALDH1A1L3MBTL1MAPTCYP1A2LMNA
SCHEMBL13701003 0.63 AURKB (0.46) ALDH1A1L3MBTL1MAPTCYP1A2MEN1
SCHEMBL21807407 0.63 PDCD1 (0.37) LMNAMEN1KMT2A
SCHEMBL21807299 0.63 KDR (0.38) ALDH1A1L3MBTL1MAPTCYP1A2LMNA
SCHEMBL21783714 0.63 KDR (0.45) ALDH1A1MAPTCYP3A4LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008057402-A2 N-ARYL-ISOXAZOLOPYRIMIDIN-4-AMINES AND RELATED COMPOUNDS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2008-05-15 WO disclosed