SCHEMBL4784756

SCHEMBL4784756

NC(=O)[C@@H]1CCCN1C(=O)c1ccccc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.51
DPP4 P27487 1/20 0.49
SPHK2 Q9NRA0 1/20 0.49
SPHK1 Q9NYA1 1/20 0.49
TRPV1 Q8NER1 1/20 0.48
FPR2 P25090 6/20 0.48
FPR1 P21462 1/20 0.48
MTTP P55157 1/20 0.47
SCN9A Q15858 2/20 0.45
HCRTR1 O43613 4/20 0.44
HCRTR2 O43614 2/20 0.43
DGAT1 O75907 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740969 0.88 PDK2 (0.51) PDK2DPP4SPHK2SPHK1TRPV1
SCHEMBL4784760 0.83 HCRTR1 (0.53) TRPV1FPR2FPR1MTTPHCRTR1
SCHEMBL3048571 0.81 RORB (0.50) PDK2TRPV1HCRTR1HCRTR2
SCHEMBL3058402 0.80 SCN9A (0.49) FPR2FPR1SCN9AHCRTR1HCRTR2
SCHEMBL3187599 0.79 GAA (0.65) TRPV1MTTPHCRTR1HCRTR2
SCHEMBL1398880 0.79 TSHR (0.54) HCRTR1HCRTR2
SCHEMBL16777183 0.79 PDK2 (0.43) PDK2SPHK2SPHK1SCN9AHCRTR1
SCHEMBL2931380 0.78 HCRTR1 (0.46) FPR2FPR1MTTPHCRTR1HCRTR2
SCHEMBL3058143 0.77 HCRTR1 (0.49) FPR2HCRTR1HCRTR2
SCHEMBL16777070 0.77 PDK2 (0.40) PDK2SPHK2SPHK1SCN9AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087611-A2 PYRROLIDINE- AND PIPERIDINE- BIS-AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-24 WO disclosed