SCHEMBL4786115

SCHEMBL4786115

Cc1c(C(=O)O)c2c(n1-c1ccccc1)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
GPR119 Q8TDV5 2/20 0.45
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
ESR2 Q92731 1/20 0.42
GRM5 P41594 2/20 0.41
GRM1 Q13255 1/20 0.41
MAPK1 P28482 1/20 0.41
NR1H2 P55055 1/20 0.41
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGDS O60760 1/20 0.39
MYC P01106 1/20 0.38
UCHL1 P09936 1/20 0.38
MAP3K14 Q99558 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789331 0.89 ADORA1 (0.51) ADORA1GPR119HDAC1HDAC6MAPT
SCHEMBL4788162 0.82 HDAC1 (0.56) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL5107551 0.81 HDAC1 (0.57) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL31078485 0.81 HDAC1 (0.57) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL4786111 0.77 GPR119 (0.46) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL28603644 0.76 BAZ2B (0.51) GPR119HDAC1HDAC6ESR2GRM5
SCHEMBL5114861 0.76 PTGDR2 (0.49) HDAC1HDAC6GRM5GRM1HPGDS
SCHEMBL968966 0.74 HDAC1 (0.50) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL4789515 0.73 MAP3K14 (0.45) ADORA1GPR119HDAC1HDAC6ESR2
SCHEMBL28602906 0.73 HDAC1 (0.54) HDAC1HDAC6ESR2GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134354-A1 TNF-α PRODUCTION INHIBITOR ARRAY BIOPHARMA, INC. (US) 2008-11-06 WO disclosed