SCHEMBL4786565

SCHEMBL4786565

CCOC(=O)[C@H](Cc1ccc(-n2c(-c3cccnc3)nc3cccnc32)cc1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 17/20 0.58
ITGB1 P05556 16/20 0.58
AKT1 P31749 1/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
PDE4B Q07343 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730881 0.93 ITGA4 (0.53) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4735439 0.90 ITGA4 (0.65) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4734610 0.83 ITGA4 (0.61) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4734486 0.82 ITGB1 (0.62) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4734787 0.82 ITGB1 (0.55) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4733969 0.81 ITGA4 (0.54) ITGA4ITGB1CYP3A4PDE4B
SCHEMBL4734732 0.81 ITGB1 (0.84) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4736515 0.79 ITGB1 (0.84) ITGA4ITGB1AKT1CYP3A4CYP2C9
SCHEMBL4733944 0.79 ITGB1 (0.84) ITGA4ITGB1CYP3A4CYP2C9
SCHEMBL4735614 0.78 ITGB1 (0.84) ITGA4ITGB1AKT1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed