SCHEMBL4787409

SCHEMBL4787409

CC(=O)N1CCCC(n2c(-c3ccccc3)c(C(=O)N3CCN(C(=O)O)CC3)[nH]c2=O)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
MAPK1 P28482 4/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
KDM6B O15054 1/20 0.35
KDM4A O75164 1/20 0.35
KDM5C P41229 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM2A Q9Y2K7 1/20 0.35
KDM3A Q9Y4C1 1/20 0.35
BTK Q06187 1/20 0.35
HSD11B1 P28845 3/20 0.34
CNR1 P21554 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL885496 0.91 SIGMAR1 (0.39) HTR2ATMEM97SIGMAR1DRD2DRD4
SCHEMBL2062636 0.88 BTK (0.44) BTKMEN1KMT2A
SCHEMBL885863 0.86 MAPK1 (0.44) DRD2DRD4DRD3MAPK1ALDH1A1
SCHEMBL885569 0.85 JAK2 (0.42) HTR2ATMEM97SIGMAR1DRD2DRD4
SCHEMBL2063261 0.79 CA1 (0.43) DRD2DRD4DRD3ALDH1A1CYP3A4
SCHEMBL2063262 0.79 CA1 (0.43) DRD2DRD4DRD3ALDH1A1CYP3A4
SCHEMBL885518 0.77 GHSR (0.39) DRD2DRD4DRD3MAPK1ALDH1A1
SCHEMBL885576 0.77 GHSR (0.39) DRD2DRD4DRD3MAPK1ALDH1A1
SCHEMBL2063126 0.77 MEN1 (0.46) MAPK1BTKMEN1KMT2A
SCHEMBL885480 0.77 JAK2 (0.41) HTR2ATMEM97SIGMAR1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089005-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-24 WO disclosed