SCHEMBL4787433

SCHEMBL4787433

O=C1COCc2cnccc21

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
AAK1 Q2M2I8 7/20 0.38
CDC25B P30305 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
ROCK2 O75116 8/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31618253 0.85 MAOA (0.38) CYP1A2CYP11B1CYP11B2MAOAMAOB
SCHEMBL4323285 0.78 CYP1A2 (0.53) CYP1A2CYP11B1CYP11B2MAOAMAOB
SCHEMBL29792666 0.78 CYP1A2 (0.53) CYP1A2CYP11B1CYP11B2MAOAMAOB
SCHEMBL147460 0.74
SCHEMBL6608536 0.74 MAOA (0.55) CYP1A2MAOAMAOBAAK1ROCK2
SCHEMBL2877256 0.74 MAOA (0.53) CYP1A2CYP11B1CYP11B2MAOAMAOB
SCHEMBL31128508 0.74 MAOA (0.53) CYP1A2CYP11B1CYP11B2MAOAMAOB
Hydrochloric Acid SCHEMBL2883050 0.73 MAOA (0.52) CYP1A2CYP11B1CYP11B2MAOAMAOB
SCHEMBL135207 0.71 MAOA (0.56) CYP1A2MAOAMAOBCDC25B
SCHEMBL29452852 0.71 MAOA (0.56) CYP1A2MAOAMAOBCDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed