SCHEMBL4787452

SCHEMBL4787452

COc1cc2cnn(C(C)=O)c2cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.54
AURKA O14965 1/20 0.54
DAPK3 O43293 1/20 0.54
CSNK1A1 P48729 1/20 0.54
GSK3A P49840 1/20 0.54
LIMK1 P53667 1/20 0.54
IKBKE Q14164 1/20 0.54
MAPK14 Q16539 1/20 0.54
TAOK1 Q7L7X3 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
DYRK1B Q9Y463 1/20 0.54
RAB9A P51151 3/20 0.45
NPC1 O15118 2/20 0.45
SHMT2 P34897 2/20 0.45
GAA P10253 2/20 0.45
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
HSP90AB1 P08238 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5407783 0.78 CHEK1 (0.49) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL19780078 0.78 CHEK1 (0.51) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL680218 0.77 CHEK1 (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL21797005 0.76 CHEK1 (0.47) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL26053980 0.76 CHEK1 (0.57) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL29288245 0.75 ALDH1A1 (0.40) RAB9ANPC1SHMT2GAACASP3
SCHEMBL18578596 0.75 HSP90AB1 (0.41) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL22359419 0.75 CHEK1 (0.43) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL16022869 0.75 MAPK14 (0.46) CHEK1AURKADAPK3CSNK1A1GSK3A
SCHEMBL5413013 0.74 CHEK1 (0.48) CHEK1AURKADAPK3CSNK1A1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089436-A2 CRYSTALLINE FORMS OF HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2008-07-24 WO disclosed
WO-2008089436-A2 CRYSTALLINE FORMS OF HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2008-07-24 WO disclosed