SCHEMBL4787688

SCHEMBL4787688

COc1ccc(-c2nc(SC)cc(N3CCOCC3)n2)cc1S(=O)(=O)N1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.53
BRD2 P25440 1/20 0.53
BRD3 Q15059 1/20 0.53
KDM4E B2RXH2 3/20 0.48
MAPT P10636 2/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
POLB P06746 1/20 0.47
SYK P43405 3/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
LMNA P02545 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4787693 0.81 CYP2C9 (0.39) BRD4BRD2BRD3KDM4EMAPT
SCHEMBL4788324 0.78 BRD4 (0.49) BRD4BRD2BRD3KDM4EMAPT
SCHEMBL7892625 0.78 BRD4 (0.49) BRD4BRD2BRD3KDM4EMAPT
SCHEMBL15120570 0.70 KMT2A (0.81) BRD4BRD2BRD3ALDH1A1MAPK1
SCHEMBL11919283 0.70 ALDH1A1 (0.68) BRD4BRD2BRD3ALDH1A1MAPK1
SCHEMBL23847020 0.69 ALDH1A1 (0.63) BRD4BRD2BRD3KDM4EALDH1A1
SCHEMBL15052436 0.69 GAA (0.77) BRD4BRD2BRD3KDM4EALDH1A1
SCHEMBL1150847 0.69 TSHR (0.75) BRD4BRD2BRD3KDM4EMAPT
SCHEMBL30511773 0.69 ALDH1A1 (0.63) BRD4BRD2BRD3KDM4EALDH1A1
SCHEMBL30511774 0.69 ALDH1A1 (0.63) BRD4BRD2BRD3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110891-A2 NEW HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED, (IN) 2008-09-18 WO claimed