SCHEMBL4787693

SCHEMBL4787693

COc1ccc(-c2nc(SC)cc(N3CCOCC3)n2)cc1S(=O)(=O)C1CNCCO1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.39
CYP1A2 P05177 4/20 0.39
CYP2C19 P33261 4/20 0.39
CYP3A4 P08684 3/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ATR Q13535 2/20 0.37
MTOR P42345 5/20 0.37
PIK3CA P42336 2/20 0.37
ADRB2 P07550 1/20 0.36
BRD4 O60885 3/20 0.36
BRD2 P25440 2/20 0.35
BRD3 Q15059 2/20 0.35
EHMT2 Q96KQ7 1/20 0.35
EHMT1 Q9H9B1 1/20 0.35
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788321 0.82 ALDH1A1 (0.37) MAPTKDM4EMTORPIK3CABRD4
SCHEMBL4787688 0.81 BRD4 (0.53) CYP2C9CYP1A2CYP2C19CYP3A4MAPT
SCHEMBL6025161 0.65 SLC6A2 (0.39)
SCHEMBL4748170 0.62 CA2 (0.46) MAPTKDM4EMTORPIK3CACA2
SCHEMBL7900089 0.62 CA2 (0.46) MAPTMTORPIK3CABRD4BRD2
SCHEMBL7892625 0.62 BRD4 (0.49) MAPTKDM4EMEN1KMT2AMTOR
SCHEMBL4788324 0.62 BRD4 (0.49) MAPTKDM4EMTORBRD4BRD2
SCHEMBL1271555 0.62 MTOR (0.64) CYP2C9CYP1A2CYP2C19MAPTKDM4E
SCHEMBL1270925 0.61 MTOR (0.67) CYP2C9CYP3A4ATRMTORPIK3CA
SCHEMBL1271916 0.59 MTOR (0.60) CYP2C9CYP1A2CYP2C19KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008110891-A2 NEW HETEROCYCLIC COMPOUNDS ORCHID RESEARCH LABORATORIES LIMITED, (IN) 2008-09-18 WO claimed