SCHEMBL4787938

SCHEMBL4787938

CC(C)(C)[Si](C)(C)OCc1cccc(CC(=O)NCCc2ccc(O)c3[nH]c(=O)sc23)c1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 17/20 0.49
ABCB11 O95342 2/20 0.41
ADRB1 P08588 1/20 0.41
DRD2 P14416 1/20 0.41
PDE4A P27815 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14099977 0.87 ADRB2 (0.54) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL4787942 0.81 ADRB2 (0.49) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL4787937 0.78 ADRB2 (0.49) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL8674037 0.76 ADRB2 (0.55) ADRB2ADRB1DRD2
SCHEMBL4739379 0.74 ADRB2 (0.53) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL27717348 0.72 ADRB2 (0.59) ADRB2ABCB11ADRB1DRD2PDE4A
Hydrochloric Acid SCHEMBL27738410 0.71 ADRB2 (0.58) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL4443114 0.70 ADRB2 (0.68) ADRB2ABCB11
SCHEMBL4440137 0.70 ADRB2 (0.56) ADRB2ABCB11ADRB1DRD2PDE4A
SCHEMBL7838985 0.70 ADRB2 (0.67) ADRB2ABCB11ADRB1DRD2PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008149110-A1 BICYCLOR [2.2.1] HEPT-7-YLAMINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASES AND CONDITIONS IN WHICH M3 MUSCARINIC RECEPTOR ACTIVITY AND BETA-ADRENERGIC ACTIVITY ARE IMPLICATED ARGENTA DISCOVERY LIMITED (GB) 2008-12-11 WO disclosed
WO-2008096127-A2 BICYCLO[2.2.1]HEPT-7-YLAMINE DERIVATIVES AND THEIR USE AS M3 MUSCARINIC RECEPTOR MODULATORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed