SCHEMBL8674037

SCHEMBL8674037

COc1ccc(CC(=O)NCCc2ccc(O)c3[nH]c(=O)sc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 11/20 0.55
ALDH1A1 P00352 2/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
POLB P06746 1/20 0.47
ERCC1 P07992 1/20 0.47
ERCC4 Q92889 1/20 0.47
ADRB1 P08588 1/20 0.47
DRD2 P14416 1/20 0.47
ADRA1D P25100 1/20 0.47
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739379 0.86 ADRB2 (0.53) ADRB2ADRB1DRD2
SCHEMBL9522342 0.85 ADRB2 (0.72) ADRB2ADRB1DRD2ADRA1D
Hydrochloric Acid SCHEMBL8882013 0.84 ADRB2 (0.71) ADRB2ADRB1DRD2ADRA1D
SCHEMBL9520760 0.82 ADRB2 (0.66) ADRB2ADRB1DRD2ADRA1D
SCHEMBL14099977 0.82 ADRB2 (0.54) ADRB2ADRB1DRD2ADRA1D
Hydrochloric Acid SCHEMBL8881126 0.82 ADRB2 (0.65) ADRB2ADRB1DRD2ADRA1D
SCHEMBL4440137 0.78 ADRB2 (0.56) ADRB2ADRB1DRD2
SCHEMBL4787938 0.76 ADRB2 (0.49) ADRB2ADRB1DRD2
SCHEMBL3685868 0.75 ADRB2 (0.49) ADRB2ADRB1DRD2
SCHEMBL14077127 0.75 ADRB2 (0.56) ADRB2ADRB1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763465-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1998-06-09 US disclosed
US-5648370-A 7-(2-aminoethyl) benzothiazolones ASTRA PHARMACEUTICALS LIMITED (GB) 1997-07-15 US disclosed
WO-1992008708-A1 BIOLOGICALLY ACTIVE AMINES FISONS PLC (GB) 1992-05-29 WO disclosed