SCHEMBL4787945

SCHEMBL4787945

CC(C)(C)[Si](C)(C)Oc1ccccc1S

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.33
CA1 P00915 5/20 0.33
CA9 Q16790 5/20 0.33
PREP P48147 2/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA7 P43166 1/20 0.31
CA14 Q9ULX7 1/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30556213 0.85 CA1 (0.38) CA12CA1CA9PREPCA2
SCHEMBL29787984 0.79 HTT (0.35) CA12CA1CA9PREPCA2
SCHEMBL11856938 0.79 CA1 (0.36) CA12CA1CA9CA2CA4
SCHEMBL29847229 0.79 CA1 (0.36) CA12CA1CA9CA2CA4
SCHEMBL24167590 0.78 CA1 (0.54) CA12CA1CA9CA2CA4
SCHEMBL30556207 0.78 TSHR (0.44) CA12CA1CA9PREP
SCHEMBL2329763 0.78 TSHR (0.44) CA12CA1CA9PREP
SCHEMBL29497318 0.78 HTR7 (0.39) CA12CA1CA9
SCHEMBL1863318 0.78 HTR7 (0.39) CA12CA1CA9
SCHEMBL2411136 0.77 ADRA2A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101029-A2 USE OF THIAZOLE, OXAZOLE AND IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-21 WO disclosed
EP-0465802-A1 Oxidant sensitive and insensitive aromatic esters as inhibitors of human neutrophil elastase CORTECH, INC. (US) 1992-01-15 EP disclosed