SCHEMBL4788079

SCHEMBL4788079

COc1cc(C2CCC(C)(CO)CC2)c(C(C)=NOCc2ccc([N+](=O)[O-])cc2)cc1O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.43
TLR3 O15455 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 4/20 0.36
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
RAB9A P51151 2/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
ALDH1A1 P00352 3/20 0.34
TTR P02766 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KLF5 Q13887 1/20 0.34
MAPK1 P28482 2/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15255527 1.00 S1PR1 (0.43) S1PR1TLR3HTTMAPTNPC1
SCHEMBL15255529 1.00 S1PR1 (0.43) S1PR1TLR3HTTMAPTNPC1
SCHEMBL10102222 0.90 S1PR1 (0.44) S1PR1TLR3HTTMAPTNPC1
SCHEMBL10102217 0.90 S1PR1 (0.44) S1PR1TLR3HTTMAPTNPC1
SCHEMBL4788191 0.89 HSP90AA1 (0.44) S1PR1TLR3HTTMAPTNPC1
SCHEMBL15255524 0.82 ALDH1A1 (0.34) HTTALDH1A1LMNA
SCHEMBL15255528 0.82 ALDH1A1 (0.34) HTTALDH1A1LMNA
SCHEMBL10101780 0.78 POLB (0.34) S1PR1MAPTL3MBTL1
SCHEMBL10101781 0.78 POLB (0.34) S1PR1MAPTL3MBTL1
SCHEMBL660122 0.78 HTT (0.43) HTTMAPTNPC1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8536157-B2 Non-steroidal compounds THE UNIVERSITY OF MELBOURNE (AU) 2013-09-17 US disclosed
WO-2008124878-A1 NON-STEROIDAL COMPOUNDS CRYPTOPHARMA PTY LTD (AU) 2008-10-23 WO disclosed