SCHEMBL4788286

SCHEMBL4788286

Cc1c(C(=O)N[C@@H]2COc3cccc(N4CCN(C)CC4)c3C2)cnn1-c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.67
SCN9A Q15858 7/20 0.67
SCN5A Q14524 5/20 0.67
TRPV4 Q9HBA0 2/20 0.48
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
ROCK2 O75116 1/20 0.42
HPGD P15428 1/20 0.42
PKM P14618 1/20 0.42
HTR1A P08908 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788603 0.91 SCN9A (0.60) KCNH2SCN9ASCN5ATRPV4MAPK1
SCHEMBL4788131 0.84 TRPV4 (0.49) KCNH2SCN9ASCN5ATRPV4NPC1
SCHEMBL4788106 0.82 SCN9A (0.73) KCNH2SCN9ASCN5ANPC1RAB9A
SCHEMBL4788881 0.80 SCN9A (0.68) KCNH2SCN9ASCN5ANPC1RAB9A
SCHEMBL20288009 0.80 SCN9A (1.00) KCNH2SCN9ASCN5APKM
SCHEMBL8075560 0.79 KCNH2 (0.61) KCNH2SCN9ASCN5A
SCHEMBL4788731 0.79 SCN9A (0.66) KCNH2SCN9ASCN5A
SCHEMBL4830493 0.77 SCN9A (0.63) KCNH2SCN9ASCN5A
SCHEMBL4830490 0.77 SCN9A (0.63) KCNH2SCN9ASCN5A
SCHEMBL4748122 0.77 SCN9A (0.65) KCNH2SCN9ASCN5AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130322-A1 NOVEL 5-HETEROCYCLYL-CHROMANE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed