SCHEMBL4788477

SCHEMBL4788477

Cc1c(C(=O)N[C@@H]2COc3cccc(N4CCN(C)CC4)c3C2)nnn1Cc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.64
KCNH2 Q12809 7/20 0.64
SCN5A Q14524 5/20 0.64
DRD2 P14416 8/20 0.52
DRD4 P21917 8/20 0.52
DRD3 P35462 8/20 0.52
HTR2A P28223 7/20 0.52
RIPK1 Q13546 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788881 0.80 SCN9A (0.68) SCN9AKCNH2SCN5ARIPK1
SCHEMBL4840071 0.78 KCNH2 (0.64) SCN9AKCNH2SCN5ADRD2DRD3
SCHEMBL4840083 0.78 KCNH2 (0.64) SCN9AKCNH2SCN5ADRD2DRD3
SCHEMBL20288009 0.78 SCN9A (1.00) SCN9AKCNH2SCN5ADRD2DRD3
SCHEMBL4789431 0.77 SCN9A (0.60) SCN9AKCNH2SCN5ARIPK1
SCHEMBL4840371 0.77 KCNH2 (0.62) SCN9AKCNH2SCN5ADRD2DRD3
SCHEMBL4840362 0.77 KCNH2 (0.62) SCN9AKCNH2SCN5ADRD2DRD3
SCHEMBL4788286 0.76 KCNH2 (0.67) SCN9AKCNH2SCN5A
SCHEMBL4748122 0.75 SCN9A (0.65) SCN9AKCNH2SCN5ADRD2DRD4
SCHEMBL4788603 0.74 SCN9A (0.60) SCN9AKCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed