SCHEMBL4789431

SCHEMBL4789431

Cc1c(C(=O)N[C@@H]2COc3cccc(N4CCN(C)CC4)c3C2)nnn1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.60
KCNH2 Q12809 7/20 0.60
SCN5A Q14524 5/20 0.60
SMN1; SMN2 Q16637 2/20 0.49
ROCK1 Q13464 1/20 0.42
CCR1 P32246 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
RIPK1 Q13546 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788710 0.86 SMN1; SMN2 (0.50) SCN9AKCNH2SCN5ASMN1; SMN2ROCK1
SCHEMBL4788881 0.80 SCN9A (0.68) SCN9AKCNH2SCN5ASMN1; SMN2MEN1
SCHEMBL4830465 0.79 SCN9A (0.80) SCN9AKCNH2SCN5A
SCHEMBL4841770 0.79 SCN9A (0.80) SCN9AKCNH2SCN5A
SCHEMBL4830458 0.79 SCN9A (0.80) SCN9AKCNH2SCN5A
SCHEMBL4830469 0.79 SCN9A (0.66) SCN9AKCNH2SCN5AMEN1KMT2A
SCHEMBL4830463 0.79 SCN9A (0.66) SCN9AKCNH2SCN5AMEN1KMT2A
SCHEMBL2079393 0.78 SMN1; SMN2 (0.62) SMN1; SMN2ROCK1CCR1KDM4EMEN1
SCHEMBL4788477 0.77 SCN9A (0.64) SCN9AKCNH2SCN5ARIPK1
SCHEMBL20288009 0.75 SCN9A (1.00) SCN9AKCNH2SCN5AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed