SCHEMBL4788975

SCHEMBL4788975

Oc1cc2c(cc1I)CCCN2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.44
KDM4E B2RXH2 4/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
ATM Q13315 1/20 0.38
GAA P10253 4/20 0.37
ALDH1A1 P00352 3/20 0.37
TP53 P04637 2/20 0.37
ALOX15 P16050 2/20 0.37
HTT P42858 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
LMNA P02545 1/20 0.37
THRB P10828 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20877573 0.84 KDM4E (0.49) MAPTKDM4ECA12CA1CA2
SCHEMBL31443901 0.78 CA12 (0.46) MAPTKDM4ECA12CA1CA2
SCHEMBL10201433 0.76 KDM4E (0.41) KDM4EALDH1A1TP53HTTLMNA
SCHEMBL21635516 0.74 MAPT (0.44) MAPTKDM4ECA12CA1CA2
SCHEMBL4788966 0.74 HTR2A (0.43) MAPTKDM4ECA12CA1CA2
SCHEMBL11317582 0.73 MAPT (0.54) MAPTKDM4EGAAALDH1A1HSD17B10
SCHEMBL9334616 0.73 MAPT (0.41) MAPTKDM4ECA12CA1CA2
SCHEMBL93915 0.71 DRD2 (0.57) MAPTKDM4EDRD2DRD4ALDH1A1
SCHEMBL15290389 0.71 MAPT (0.47) MAPTKDM4ECA12CA1CA2
SCHEMBL29358285 0.71 DRD2 (0.57) MAPTKDM4EDRD2DRD4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632261-B1 INHIBITORS OF HEPATITIS C VIRUS PRESIDIO PHARMACEUTICALS INC (US) 2016-07-13 EP disclosed
WO-2012058125-A1 INHIBITORS OF HEPATITIS C VIRUS PRESIDIO PHARMACEUTICALS, INC. (US) 2012-05-03 WO disclosed