SCHEMBL4789142

SCHEMBL4789142

O=C1NC(=O)C(c2ccc(OC=S)cc2)=C1c1ccc(O)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.51
GSK3B P49841 6/20 0.42
SENP1 Q9P0U3 1/20 0.39
ESR2 Q92731 2/20 0.38
ESR1 P03372 1/20 0.38
GSK3A P49840 1/20 0.36
AKR1B1 P15121 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NAT1 P18440 1/20 0.36
PREP P48147 1/20 0.35
ME2 P23368 1/20 0.34
ME1 P48163 1/20 0.34
ME3 Q16798 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788888 0.85 PTGS2 (0.50) PTGS2GSK3BHPGDNAT1
SCHEMBL4460171 0.78 MEN1 (0.50) PTGS2ESR2ESR1HPGDRAB9A
SCHEMBL6702892 0.71 PTGS2 (0.59) PTGS2GSK3BSENP1ESR2ESR1
SCHEMBL9065257 0.68 PTGS2 (0.61) PTGS2GSK3BSENP1ESR2ESR1
SCHEMBL28862647 0.68 GSK3B (0.57) PTGS2GSK3BSENP1ESR2ESR1
SCHEMBL14026490 0.68 PTGS2 (0.56) PTGS2GSK3BSENP1ESR2ESR1
SCHEMBL28080907 0.67 PTGS2 (0.72) PTGS2GSK3BGSK3ARAB9ATDP1
SCHEMBL4752018 0.67 PTGS2 (0.49) PTGS2HPGDTDP1
SCHEMBL18049411 0.67 PTGS2 (0.54) PTGS2GSK3BSENP1ESR2ESR1
SCHEMBL22954264 0.66 ESR2 (0.58) PTGS2GSK3BESR2ESR1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO claimed
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO disclosed